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Products Details
Product Description
– MS012 is a selective GLP inhibitor (IC50=7 nM). MS012 can be used in research of GLP dysregulation, including cancer, inflammatory diseases, and neuroregenerative disorders[1].
Web ID
– HY-114628
Shipping
– Room temperature
Molecular Formula
– C22H35N5O2
References
– [1]Xiong Y, et al. Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase. J Med Chem. 2017 Mar 9;60(5):1876-1891.
CAS Number
– 2089617-83-2
Molecular Weight
– 401.55
SMILES
– COC1=CC2=NC(NCCCCCC)=NC(NC3CCN(CC3)C)=C2C=C1OC
Clinical Information
– No Development Reported
Research Area
– Cancer; Inflammation/Immunology; Neurological Disease
Solubility
– 10 mM in DMSO
Target
– GLP Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
