LSN2814617
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LSN2814617

SKU T27855-25 mg Category Brand:

Price range: 2,432 CAD through 4,000 CAD

Products Details

Product Description

– LSN2814617 is an orally active, potent, brain-penetrant, and selective mGlu 5 (metabotropic glutamate 5) positive allosteric modulator (PAM), with EC 50 values of 52 nM (Human mGlu5) and 42 nM (rat mGlu5). In vivo EEG studies demonstrated that LSN2463359 has marked wake-promoting properties with minimal rebound hypersomnolence, and it can be used for schizophrenia research [1].

Web ID

– T27855

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C18H20FN5O

References

– Loomis S, McCarthy A, Baxter C, Kellett DO, Edgar DM, Tricklebank M, Gilmour G. Distinct pro-vigilant profile induced in rats by the mGluR5 potentiator LSN2814617. Psychopharmacology (Berl). 2015 Nov;232(21-22):3977-89. doi: 10.1007/s00213-015-3936-8. PubMed PMID: 25902875; PubMed Central PMCID: PMC4600478.

CAS Number

– 1313498-17-7

Molecular Weight

– C18H20FN5O

SMILES

– C(C)(C)(C)C=1N2C(C[C@H](CC2)C3=NC(=NO3)C4=CC=C(F)C=C4)=NN1

Pathway

– Others

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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