K-Opioid receptor agonist-1

SKU T88205-25 mg Category Brand:

Price range: 4,112 CAD through 7,360 CAD

Products Details

Product Description

– K-Opioid receptor agonist-1 (Compound 5a) acts as an agonist for the κ-Opioid receptor, exhibiting a K_i of 0.25 nM and an EC_50 of 2 nM. This compound is capable of crossing the blood-brain barrier (BBB), evidenced by brain/plasma ratios ranging from 0.50 to 0.65. Additionally, K-Opioid receptor agonist-1 demonstrates anti-inflammatory effects in dermatitis models induced by either Arachidonic acid or oxazolidinone.

Web ID

– T88205

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C22H29Cl2N3O3

CAS Number

– 1816990-29-0

Molecular Weight

– C22H29Cl2N3O3

SMILES

– C(CC1=CC(Cl)=C(Cl)C=C1)(=O)N2[C@]3([C@@](N(C(OC)=O)CC2)(CCC[C@@H]3N4CCCC4)[H])[H]

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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