GSK2656157
Add to CompareAdded to Compare

Download Files:

GSK2656157

SKU T2654-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 48 CAD through 1,064 CAD

Products Details

Product Description

– GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay. The selectivty is 500-fold higher against a panel of 300 kinases.

Web ID

– T2654

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C23H21FN6O

Citations

– 1. Tan M, Wang H, Gao C, et al. Agonists Specific for κ-Opioid Receptor Induces Apoptosis of HCC Cells Through Enhanced Endoplasmic Reticulum Stress. Frontiers in Oncology. 2022.12 2. Lu Y, Li D, Ai H, et al.Glucose-regulated protein 94 facilitates the proliferation of the Bombyx mori nucleopolyhedrovirus via inhibiting apoptosis.International Journal of Biological Macromolecules.2023: 127158. 3. Wang X, Xue Y, Hao K, et al.Sustained therapeutic effects of self-assembled hyaluronic acid nanoparticles loaded with α-Ketoglutarate in various osteoarthritis stages.Biomaterials.2025, 314: 122845.

References

– Atkins C, et al. Cancer Res, 2013, 73(6), 1993-2002.

CAS Number

– 1337532-29-2

Molecular Weight

– C23H21FN6O

Compound Purity

– 0.998

SMILES

– Cc1cccc(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1

Pathway

– Apoptosis|||Autophagy

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

Related Products

Select options
Mexenone
Mexenone Price range: 48 CAD through 157 CAD
1 mL * 10 mM (in DMSO)100 mg200 mg

1000 in stock

Select options
Flubendazole
Flubendazole Price range: 53 CAD through 149 CAD
1 mL * 10 mM (in DMSO)100 mg50 mg

1000 in stock

Select options
7-Chloro-4-(piperazin-1-yl)quinoline
7-Chloro-4-(piperazin-1-yl)quinoline Price range: 56 CAD through 77 CAD
100 mg200 mg

1000 in stock

Select options
Jedi2
Jedi2 Price range: 53 CAD through 1,117 CAD
1 mg1 mL * 10 mM (in DMSO)5 mg

1000 in stock

Select options
4-Methoxycoumarine
4-Methoxycoumarine Price range: 56 CAD through 266 CAD
1 g1 mL * 10 mM (in DMSO)50 mg

1000 in stock

My Cart
Wishlist
Recently Viewed
Categories

Request Data Sheet / Safty Data Sheet

Please enable JavaScript in your browser to complete this form.
=

Price Request

Please enable JavaScript in your browser to complete this form.
=

Compare Products (0 Products)
document.addEventListener('elementor/popup/show', function() { if (typeof turnstile !== 'undefined') { document.querySelectorAll('.cf-turnstile').forEach(function(el) { if (!el.dataset.rendered) { turnstile.render(el); el.dataset.rendered = true; } }); } });