Grp94 Inhibitor-1
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Grp94 Inhibitor-1

SKU T7261-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 66 CAD through 618 CAD

Products Details

Product Description

– Grp94 Inhibitor-1 is a potent and selective inhibitor of Grp94 with an IC50 of 2 nM.

Web ID

– T7261

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C22H28N2O2

Citations

– 1. Hao M, Guo Y, Zhang Z, et al. 6-acrylic phenethyl ester-2-pyranone derivative induces apoptosis and G2/ M arrest by targeting GRP94 in colorectal cancer. Bioorganic Chemistry. 2022, 123: 105802 2. Lu Y, Li D, Ai H, et al.Glucose-regulated protein 94 facilitates the proliferation of the Bombyx mori nucleopolyhedrovirus via inhibiting apoptosis.International Journal of Biological Macromolecules.2023: 127158.

References

– Jiang F , Guo A P , Xu J C , et al. Discovery of a Potent Grp94 Selective Inhibitor with Anti-inflammatory Efficacy in a Mouse Model of Ulcerative Colitis[J]. Journal of Medicinal Chemistry, 2018.

CAS Number

– 2234897-35-7

Molecular Weight

– C22H28N2O2

Compound Purity

– 0.9702

SMILES

– CC(C)c1ccc(cc1)-c1ccc(N[C@H]2CC[C@H](O)CC2)c(c1)C(N)=O

Pathway

– Cytoskeletal Signaling|||GPCR/G Protein|||Metabolism|||Endocrinology/Hormones

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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