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FEMA 4809
SKU
HY-130074-10 mg
Category Reference compound
Tags Membrane Transporter/Ion Channel;Neuronal Signaling, Neurological Disease, TRP Channel
$250 – $1,950
Products Details
Product Description
– FEMA 4809 is a TRPM8 receptor agonist (EC50=0.2 nM) for use as a cooling agent. TRPM8 is the ion channel responsible for the cool perception[1].
Web ID
– HY-130074
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C17H17N3O2S
References
– [1]Alain Noncovich, et al. Discovery and development of a novel class of phenoxyacetyl amides as highly potent TRPM8 agonists for use as cooling agents. Bioorg Med Chem Lett. 2017 Aug 15;27(16):3931-3938.
CAS Number
– 1374760-95-8
Molecular Weight
– 327.40
Compound Purity
– 99.25
SMILES
– O=C(N(C1=NNC=C1)CC2=CC=CS2)COC3=CC=C(C)C=C3
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– DMSO : 250 mg/mL (ultrasonic)
Target
– TRP Channel
Pathway
– Membrane Transporter/Ion Channel;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.