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Products Details
Product Description
– ERK-IN-2 free base is a ERK2 inhibitor with an IC50 value of 1.8 nM. ERK-IN-2 free base might lead to off-target toxicity and/or off-target activity at dose >10 μM[1].
Web ID
– HY-133084A
Shipping
– Room temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C16H17N5O2
References
– [1]MRK-ERK Inhibitor and Negative Control.
CAS Number
– 2743576-55-6
Molecular Weight
– 311.34
SMILES
– OCC1=C2C(NN=C2)=CC(NC(N[C@@H](C3=CC=CC=C3)C)=O)=N1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– ERK
Isoform
– ERK2
Pathway
– MAPK/ERK Pathway;Stem Cell/Wnt
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
