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EP2 receptor antagonist-1
SKU
HY-145684-10 mg
Category Reference compound
Tags GPCR/G Protein, Inflammation/Immunology, Prostaglandin Receptor
$400 – $3,400
Products Details
Product Description
– EP2 receptor antagonist-1 (compound 1) is a potent, reversible, and agonist dependent allosteric prostaglandin EP2 receptor antagonist. EP2 receptor antagonist-1 shows anti-inflammatory effects[1].
Web ID
– HY-145684
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C24H22N4O5
References
– [1]Jiang C, et, al. An Agonist Dependent Allosteric Antagonist of Prostaglandin EP2 Receptors. ACS Chem Neurosci. 2020 May 20;11(10):1436-1446.
CAS Number
– 848920-08-1
Molecular Weight
– 446.46
Compound Purity
– 99.45
SMILES
– O=C(C1=C(N)N(C2=CC=C3OCCOC3=C2)C4=C1N=C5C=CC=CC5=N4)OCC6OCCC6
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– Prostaglandin Receptor
Isoform
– EP
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.