Download Files:
Products Details
Product Description
– Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.
Web ID
– TP1931
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C79H109N19O12
References
– Holst et al (2003) High constitutive signaling of the ghrelin receptor – identification of a potent inverse agonist. Mol.Endocrinol. 17 2201 PMID:
CAS Number
– 96736-12-8
Molecular Weight
– C79H109N19O12
SMILES
– C([C@H](C(N[C@H](C(N[C@H](CC=1C=2C(NC1)=CC=CC2)C(N[C@H](C(N[C@@H](CC(C)C)C(N)=O)=O)CC(C)C)=O)=O)CC3=CC=CC=C3)=O)NC([C@@H](NC([C@H](NC(=O)[C@H]4N(C([C@@H](NC(=O)[C@H]5N(C([C@@H](CCCNC(=N)N)N)=O)CCC5)CCCCN)=O)CCC4)CC6=CC=CC=C6)=O)CCC(N)=O)=O)C=7C=8C(NC7)=CC=CC8
Product type
– Peptide
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
Related Products
Degarelix acetate(214766-78-6 free base)
112 CAD – 1,579 CADPrice range: 112 CAD through 1,579 CAD
1000 in stock
1000 in stock
1000 in stock

