Download Files:
Products Details
Product Description
– CCR2 antagonist 1 is a high-affinity antagonist of CCR2 with a Ki of 2.4 nM and a long residence time.
Web ID
– T10711
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C28H32BrF3N2O
References
– Vilums M, et al. When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists. Eur J Med Chem. 2015 Mar 26;93:121-34.
CAS Number
– 1683534-96-4
Molecular Weight
– C28H32BrF3N2O
SMILES
– CC(C)[C@@]1(CC[C@H](C1)N[C@@H]1CCc2cc(Br)ccc12)C(=O)N1CCc2ccc(cc2C1)C(F)(F)F
Target
– Potassium Channel|||Dopamine Receptor
Pathway
– GPCR/G Protein|||Immunology/Inflammation|||Microbiology/Virology
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
Related Products
1000 in stock
1000 in stock
1000 in stock
