CBP/p300-IN-5

SKU HY-100132-5 mg Category Tags , ,

$878

Only 1000 item(s) left in stock.

Products Details

Product Description

– P300/CBP-IN-5 is a potent p300/CBP histone acetyltransferase inhibitor extracted from patent WO2016044770A1, Example 715, has an IC50 of 18.8 nM[1].

Web ID

– HY-100132

Shipping

– Room temperature

Applications

– Cancer-programmed cell death

Molecular Formula

– C29H27F5N6O4

References

– [1]Michael Michaelides, et al. Spirocyclic hat inhibitors and methods for their use. WO2016044770A1.

CAS Number

– 1889284-33-6

Molecular Weight

– 618.55

SMILES

– O=C(CN(C1=O)C(N[C@@]21C[C@H](C3=C2C=CC(C4=CN(N=C4)CC(NC)=O)=C3)F)=O)N([C@H](C(F)(F)F)C)CC5=CC=C(C=C5)F

Clinical Information

– No Development Reported

Research Area

– Cancer

Solubility

– 10 mM in DMSO

Target

– Histone Acetyltransferase

Isoform

– CBP/p300

Pathway

– Epigenetics

Product type

– Reference compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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