CB2R PAM
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CB2R PAM

SKU T37075-1 mg Category Brand:

Price range: 51  USD through 1,380  USD

Products Details

Product Description

– CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTPγS binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.

Web ID

– T37075

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C21H24BrFN2O2

References

– Gado F, et al. Identification of the First Synthetic Allosteric Modulator of the CB2 Receptors and Evidence of Its Efficacy for Neuropathic Pain Relief. J Med Chem. 2019;62(1):276-287.

CAS Number

– 2244579-87-9

Molecular Weight

– C21H24BrFN2O2

Compound Purity

– 0.9817

SMILES

– N(C(=O)C1CCCCCC1)C=2C(=O)N(CC3=CC=C(F)C=C3)C=C(Br)C2C

Pathway

– GPCR/G Protein

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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