– 1. Dai W, Wu J, Peng X, et al. CDK12 orchestrates super‐enhancer‐associated CCDC137 transcription to direct hepatic metastasis in colorectal cancer. Clinical and Translational Medicine. 2022, 12(10): e1087. 2. Yang X, Cheng B, Xiao Y, et al. Discovery of Novel CA-4 Analogs as Dual Inhibitors of Tubulin Polymerization and PD-1/PD-L1 Interaction for Cancer Treatment. European Journal of Medicinal Chemistry. 2021 Mar 5;213:113058. doi: 10.1016 3. Zhang H, Zhou S, Plewka J, et al.Design, Synthesis, and Antitumor Activity Evaluation of 2-Arylmethoxy-4-(2, 2′-dihalogen-substituted biphenyl-3-ylmethoxy) Benzylamine Derivatives as Potent PD-1/PD-L1 Inhibitors.Journal of Medicinal Chemistry.2023 4. Zhang H, Zhou S J, Shen C F, et al.PD-L1 dimerisation induced by biphenyl derivatives mediates anti-breast cancer activity via the non-immune PD-L1–AKT–mTOR/Bcl2 pathway.Journal of Enzyme Inhibition and Medicinal Chemistry.2023, 38(1): 2230388. 5. Zhang F, Zhang H, Zhou S, et al.Design, synthesis, and evaluation of antitumor activity of 2-arylmethoxy-4-(2-fluoromethyl-biphenyl-3-ylmethoxy) benzylamine derivatives as PD-1/PD-L1 inhibitors.European Journal of Medicinal Chemistry.2024: 116683.