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Aticaprant
Price range: 54 CAD through 1,022 CAD
Products Details
Product Description
– Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).[2]
Web ID
– TQ0082
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C26H27FN2O2
References
– Rorick-Kehn LM, et al. LY2456302 is a novel, potent, orally-bioavailable small molecule kappa-selective antagonist with activity in animal models predictive of efficacy in mood and addictive disorders. Neuropharmacology. 2014 Feb;77:131-44.
CAS Number
– 1174130-61-0
Molecular Weight
– C26H27FN2O2
Compound Purity
– 0.9993
SMILES
– Cc1cc(C)cc(c1)[C@@H]1CCCN1Cc1ccc(Oc2ccc(cc2F)C(N)=O)cc1
Pathway
– Endocrinology/Hormones|||Neuroscience|||GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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