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Asapiprant
SKU
HY-16763-1 mg
Category Reference compound
Tags GPCR/G Protein, Inflammation/Immunology; Endocrinology, Prostaglandin Receptor
$165 – $3,245
Products Details
Product Description
– Asapiprant is a potent and selective DP1 receptor antagonist with a Ki of 0.44 nM.
Web ID
– HY-16763
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C24H27N3O7S
References
– [1]Takahashi G, et al. Effect of the potent and selective DP1 receptor antagonist, asapiprant (S-555739), in animal models of allergic rhinitis and allergic asthma. Eur J Pharmacol. 2015 Oct 15;765:15-23.
CAS Number
– 932372-01-5
Molecular Weight
– 501.55
Compound Purity
– 99.53
SMILES
– O=C(O)COC1=CC(N2CCN(S(=O)(C3=CC=C(OC(C)C)C=C3)=O)CC2)=CC=C1C4=NC=CO4
Clinical Information
– Phase 2
Research Area
– Inflammation/Immunology; Endocrinology
Solubility
– DMSO : 11.11 mg/mL (ultrasonic)
Target
– Prostaglandin Receptor
Isoform
– DP
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.