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Product Description
– Apelin agonist 1 is an oral selective apelin agonist AM-2995, a agonist of the APJ (APLNR, angiotensin receptor like-1) receptor, may be used in the treatment of cardiovascular conditions. Apelin agonist 1 is extracted from patent WO 2018097944 (210.0), Example 210.0[1].
Web ID
– HY-126293
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C23H20FN5O5S
References
– [1]Matthew Brown, et al. Triazole furan compounds as agonists of the apj receptor
CAS Number
– 2227512-85-6
Molecular Weight
– 497.50
SMILES
– O=S(CCC1=CC=C(F)C=C1C#N)(NC2=NN=C(C3=CC=CO3)N2C4=C(OC)C=CC=C4OC)=O
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– Apelin Receptor (APJ)
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
