Aticaprant

SKU TQ0082-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 54 CAD through 1,022 CAD

Products Details

Product Description

– Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).[2]

Web ID

– TQ0082

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C26H27FN2O2

References

– Rorick-Kehn LM, et al. LY2456302 is a novel, potent, orally-bioavailable small molecule kappa-selective antagonist with activity in animal models predictive of efficacy in mood and addictive disorders. Neuropharmacology. 2014 Feb;77:131-44.

CAS Number

– 1174130-61-0

Molecular Weight

– C26H27FN2O2

Compound Purity

– 0.9993

SMILES

– Cc1cc(C)cc(c1)[C@@H]1CCCN1Cc1ccc(Oc2ccc(cc2F)C(N)=O)cc1

Pathway

– Endocrinology/Hormones|||Neuroscience|||GPCR/G Protein

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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