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MEN 11270
429 CAD
Only 1000 item(s) left in stock.
Products Details
Product Description
– Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3); conformationally constrained cyclized analog of HOE 140. Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other receptors and ion channels (pIC50 < 5.5).
Web ID
– TP1999
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C60H90N20O11S
References
– Meini et al (1999) MEN 11270, a novel selective constrained peptide antagonist with high affinity at the human B2 kinin receptor. J.Pharmacol.Exp.Ther. 289 1250 PMID:
CAS Number
– 235082-52-7
Molecular Weight
– C60H90N20O11S
SMILES
– O=C1N2[C@@]3([C@](C[C@]2(C(=O)N[C@@H](CCCNC(=N)N)C(=O)NCC[C@H](NC([C@H](CC4=CC=CS4)NC(CNC(=O)[C@H]5N(C(=O)[C@H]6N(C([C@@H](NC([C@@H](CCCNC(=N)N)N)=O)CCCNC(=N)N)=O)CCC6)C[C@H](O)C5)=O)=O)C(=O)N7[C@@]1(CC=8C(C7)=CC=CC8)[H])[H])(CCCC3)[H])[H]
Product type
– Peptide
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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