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[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Price range: 229 CAD through 4,784 CAD
Products Details
Product Description
– [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.
Web ID
– TP1931L1
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C81H113N19O14
References
– Holst et al (2003) High constitutive signaling of the ghrelin receptor – identification of a potent inverse agonist. Mol.Endocrinol. 17 2201 PMID:
Molecular Weight
– C81H113N19O14
Compound Purity
– 0.9768
SMILES
– CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=CNC5=C4C=CC=C5)NC([C@H](CCC(N)=O)NC([C@@H](CC6=CC=CC=C6)NC([C@H]7N(C([C@H](CCCCN)NC([C@H]8N(C([C@@H](CCCNC(N)=N)N)=O)CCC8)=O)=O)CCC7)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
Pathway
– GPCR/G Protein
Product type
– Peptide
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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