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Product Description
– α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM. It promotes the proteasomal degradation of the α1A-AR and exhibits anti-proliferative effects against PC-3 cells, presenting an IC50 value of 6.12 μM. This compound demonstrates antitumor activity and holds potential for prostate cancer research [1].
Web ID
– T74557
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C38H43N11O11
CAS Number
– 2863635-02-1
Molecular Weight
– C38H43N11O11
SMILES
– N(C(COCCOCCOCCN1C=C(C(=O)N2CCN(CC2)C3=NC4=C(C(N)=N3)C=C(OC)C(OC)=C4)N=N1)=O)C5=C6C(C(=O)N(C6=O)C7C(=O)NC(=O)CC7)=CC=C5
Pathway
– PROTAC
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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