Relugolix
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Relugolix

SKU T3630-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 59 CAD through 1,096 CAD

Products Details

Product Description

– Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively binds to and blocks the GnRH receptor in the anterior pituitary gland, which both prevents GnRH binding to the GnRH receptor and inhibits the secretion and release of both luteinizing hormone (LH) and follicle stimulating hormone (FSH). In males, the inhibition of LH secretion prevents the release of testosterone from Leydig cells in the testes. Since testosterone is required to sustain prostate growth, reducing testosterone levels may inhibit hormone-dependent prostate cancer cell proliferation.

Web ID

– T3630

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C29H27F2N7O5S

References

– MacLean DB et al. J Clin Endocrinol Metab. 2015 Dec;100(12):4579-87.

CAS Number

– 737789-87-6

Molecular Weight

– C29H27F2N7O5S

Compound Purity

– 0.9997

SMILES

– CONC(=O)Nc1ccc(cc1)-c1sc2n(Cc3c(F)cccc3F)c(=O)n(-c3ccc(OC)nn3)c(=O)c2c1CN(C)C

Target

– Cholecystokinin Receptor

Pathway

– GPCR/G Protein

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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