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ZEN-3862
Price range: 56 CAD through 949 CAD
Products Details
Product Description
– ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
Web ID
– T13394
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C19H17FN2O3
References
– Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.
CAS Number
– 1952264-33-3
Molecular Weight
– C19H17FN2O3
Compound Purity
– 0.971
SMILES
– CC=1C(C2=CN(CC3=CC(F)=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1
Target
– p53|||Ferroptosis|||Aryl Hydrocarbon Receptor
Pathway
– Chromatin/Epigenetic
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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