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(R)-Elagolix
Price range: 51 CAD through 1,171 CAD
Products Details
Product Description
– (R)-Elagolix (NBI-56418) is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
Web ID
– T11174
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C32H30F5N3O5
References
– Carr B, et al. Elagolix, an oral GnRH antagonist, versus subcutaneous depot medroxyprogesterone acetate for the treatment of endometriosis: effects on bone mineral density. Reprod Sci. 2014 Nov;21(11):1341-1351.
CAS Number
– 834153-87-6
Molecular Weight
– C32H30F5N3O5
Compound Purity
– 0.9763
SMILES
– [H][C@@](Cn1c(=O)c(c(C)n(Cc2c(F)cccc2C(F)(F)F)c1=O)-c1cccc(OC)c1F)(NCCCC(O)=O)c1ccccc1
Target
– Autophagy
Pathway
– GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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