(E)-GABAB receptor antagonist 1
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(E)-GABAB receptor antagonist 1

SKU T11137-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 187 CAD through 2,448 CAD

Products Details

Product Description

– (E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist that decreases GABA-induced IP3 (inositol trisphosphate) production with an IC50 of 37.9 μM. It is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors.

Web ID

– T11137

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C18H24O4

References

– Chen LH, et al. Discovery of a Negative Allosteric Modulator of GABAB Receptors. ACS Med Chem Lett. 2014 May 27;5(7):742-7.

CAS Number

– 1611483-29-4

Molecular Weight

– C18H24O4

Compound Purity

– 0.9526

SMILES

– C(=C/C(C(O)=O)=O)C1=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C1

Target

– Others

Pathway

– Membrane transporter/Ion channel|||Neuroscience

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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