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Tenalisib R Enantiomer
$190 – $2,200
Products Details
Product Description
– Tenalisib R Enantiomer (RP6530 R Enantiomer) is an R enantiomer of Tenalisib. Tenalisib is a potent and selective PI3Kδ and PI3Kγ inhibitor with IC50 values of 25 and 33 nM, respectively[1][2].
Web ID
– HY-112172
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C23H18FN5O2
References
– [1]Swaroop Vakkalanka, et al. Abstract 2704: RP6530, a dual PI3K δ/γ inhibitor, potentiates ruxolitinib activity in the JAK2-V617F mutant erythroleukemia cell lines.
CAS Number
– 1639417-54-1
Molecular Weight
– 415.42
Compound Purity
– 98.0
SMILES
– O=C1C(C2=CC=CC(F)=C2)=C([C@H](NC3=C4N=CNC4=NC=N3)CC)OC5=CC=CC=C15
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– PI3K
Pathway
– PI3K/Akt/mTOR
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
