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Telaglenastat
Price range: 51 CAD through 1,904 CAD
Products Details
Product Description
– Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.
Web ID
– T6797
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C26H24F3N7O3S
Citations
– 1. Caiola E, Colombo M, Sestito G, et al. Glutaminase Inhibition on NSCLC Depends on Extracellular Alanine Exploitation. Cells. 2020, 9(8): 1766
2. Zhao G, Zhu H, Xue X, et al.Feline Calicivirus Infection Manipulates Central Carbon Metabolism.Veterinary Sciences.2025, 12(2): 138.
References
– Gross MI, et al. Antitumor activity of the glutaminase inhibitor CB-839 in triple-negative breast cancer. Mol Cancer Ther. 2014 Apr;13(4):890-901.
CAS Number
– 1439399-58-2
Molecular Weight
– C26H24F3N7O3S
Compound Purity
– 0.9989
SMILES
– FC(F)(F)Oc1cccc(CC(=O)Nc2ccc(CCCCc3nnc(NC(=O)Cc4ccccn4)s3)nn2)c1
Pathway
– Autophagy|||Metabolism|||Proteases/Proteasome
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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