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TAK-448
Price range: 194 CAD through 590 CAD
Products Details
Product Description
– TAK-448 (MVT-602), a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM, has been studied in trials for the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.
Web ID
– TP1094
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C58H80N16O14
References
– Nishizawa N, et al. Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH2 (TAK-448), with Highly PotentTestosterone-Suppressive Activity and Excellent Water Solubility. J Med Chem. 2016 Oct 13;59(19):8804-8811.
CAS Number
– 1234319-68-6
Molecular Weight
– C58H80N16O14
SMILES
– C([C@H](NC([C@@H](NC([C@@H](NC(NNC([C@H](CC1=CC=CC=C1)NC([C@@H](NC([C@@H](NC(=O)[C@H]2N(C([C@@H](CC3=CC=C(O)C=C3)NC(C)=O)=O)C[C@H](O)C2)CC(N)=O)=O)[C@@H](C)O)=O)=O)=O)CC(C)C)=O)CCCNC(NC)=N)=O)C(N)=O)C=4C=5C(NC4)=CC=CC5
Product type
– Peptide
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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