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Products Details
Product Description
– StRIP16, bioavailable StRIP3 analogue, is a double-stapled peptide which can bind to Rab8a GTPase, with a Kd of 12.7 μM[1].
Web ID
– HY-136197
Shipping
– Room temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C116H154N24O26
References
– [1]Cromm PM, et, al. Protease-Resistant and Cell-Permeable Double-Stapled Peptides Targeting the Rab8a GTPase. ACS Chem Biol. 2016 Aug 19;11(8):2375-82.
CAS Number
– 2761279-63-2
Molecular Weight
– 2300.65
SMILES
– CC(C)C[C@H](NC([C@H](CC1=CN=CN1)NC([C@H](CC2=CC=C(O)C=C2)NC([C@]3(C)CCC/C=C/CCC[C@](C(N[C@@H](CCC(N)=O)C(N[C@@H](CC4=CNC5=CC=CC=C45)C(N[C@@H](CC6=CC=CC=C6)C(N3)=O)=O)=O)=O)(C)NC([C@H](CCC(O)=O)NC([C@H](CC(N)=O)NC([C@@H](NC(C)=O)CC(O)=O)=O)=O)=O)=O)=O)=O)C(N[C@@]7(C)CCC/C=C/CCC[C@](C(N[C@@H](C(C)C)C(N)=O)=O)(C)NC([C@H](CC(N)=O)NC([C@H](CC8=CC=CC=C8)NC([C@H](CC9=CC=CC=C9)NC7=O)=O)=O)=O)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Ras
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
