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Products Details
Product Description
– Risperidone E-oxime is an impurity of Risperidone[1]. Risperidone is a serotonin 5-HT2 receptor blocker, P-Glycoprotein inhibitor and potent dopamine D2 receptor antagonist, with Kis of 4.8, 5.9 nM for 5-HT2A and dopamine D2 receptor, respectively [2][3].
Web ID
– HY-135194
Shipping
– Room temperature
Molecular Formula
– C23H28F2N4O2
References
– [1]Pavel Slanina, et al. Process for making risperidone and intermediates therefor. US20040097523A1.|[2]Nyberg S, et al. 5-HT2 and D2 dopamine receptor occupancy in the living human brain. A PET study with risperidone. Psychopharmacology (Berl). 1993;110(3):265-72.|[3]Zhu HJ, et al. Risperidone and paliperidone inhibit p-glycoprotein activity in vitro. Neuropsychopharmacology. 2007 Apr;32(4):757-64.
CAS Number
– 691007-09-7
Molecular Weight
– 430.49
SMILES
– O=C1C(CCN2CCC(/C(C3=CC=C(F)C=C3F)=NO)CC2)=C(C)N=C4N1CCCC4
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– 10 mM in DMSO
Target
– Drug Metabolite
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
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