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NNC052090
Price range: 2,432 CAD through 4,000 CAD
Products Details
Product Description
– NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 μM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at α1- and D2-receptors with IC50 values are 266 and 1632 nM respectively.
Web ID
– T28183
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C27H30N2O2
References
– Dalby NO, Thomsen C, Fink-Jensen A, Lundbeck J, Søkilde B, Man CM, Sørensen PO, Meldrum B. Anticonvulsant properties of two GABA uptake inhibitors NNC 05-2045 and NNC 05-2090, not acting preferentially on GAT-1. Epilepsy Res. 1997 Jul;28(1):51-61. PubMed PMID: 9255599.
CAS Number
– 184845-43-0
Molecular Weight
– C27H30N2O2
SMILES
– C(CCN1CCC(O)(CC1)C2=C(OC)C=CC=C2)N3C=4C(C=5C3=CC=CC5)=CC=CC4
Pathway
– Others
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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