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Products Details
Product Description
– MC2652 (compound 1a) is a potent LSD1 inhibitor. MC2652 displays high inhibiting effects in MV4-11 and NB4 leukaemia cells. MC2652 shows antiproliferative activity against prostate cancer LNCaP cells[1].
Web ID
– HY-144755
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C22H20N2O
References
– [1]Fioravanti R, et al. Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity. J Enzyme Inhib Med Chem. 2022 Dec;37(1):973-985.
CAS Number
– 2771425-46-6
Molecular Weight
– 328.41
SMILES
– NC1CC1C2=CC=C(C=C2)NC(C3=CC=C(C=C3)C4=CC=CC=C4)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Demethylase
Isoform
– KDM1/LSD1
Pathway
– Epigenetics
Product type
– Reference compound
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