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GPR81 agonist 1
Price range: 211 CAD through 2,544 CAD
Products Details
Product Description
– GPR81 agonist 1 is a potent and selective GPR81 agonist with high affinity for human and mouse GPR81, inhibiting lipolysis of differentiated 3T3-L1 adipocytes, improving insulin sensitivity and glycaemic control in mouse models of insulin resistance and diabetes, and can be used in the study of diabetes and obesity.
Web ID
– T62656
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C22H30N4O2S2
References
– Sakurai T, et al. Identification of a novel GPR81-selective agonist that suppresses lipolysis in mice without cutaneous flushing. Eur J Pharmacol. 2014;727:1-7.
CAS Number
– 1620992-67-7
Molecular Weight
– C22H30N4O2S2
Compound Purity
– 0.9968
SMILES
– C[C@H]1CC[C@@H](CC1)C(=O)Nc1nc(c(CC(=O)N2CCN(C)CC2)s1)-c1cccs1
Pathway
– Endocrinology/Hormones|||GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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