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GDC-2992
Price range: 542 CAD through 6,640 CAD
Products Details
Product Description
– GDC-2992 is a selective and oral AR (androgen receptor) degrader that inhibits the proliferation of tumor cells overexpressing AR, degrades AR (DC50 = 2.7 nM) and inhibits proliferation (IC50 = 9.7 nM) in VCaP cells, and can be used for oncology studies in denuded resistant prostate cancer (CRPC).
Web ID
– T204088
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C45H51ClN8O5
CAS Number
– 2753651-10-2
Molecular Weight
– C45H51ClN8O5
Compound Purity
– 0.9982
SMILES
– O([C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(C=C2)N3CCC(CN4CCN(CC4)C=5C=C6C(=CC5)C(=O)N(N=C6)[C@@H]7C(=O)NC(=O)CC7)CC3)C1(C)C)C8=CC(Cl)=C(C#N)C=C8
Target
– Monoamine Oxidase
Pathway
– PROTAC|||Endocrinology/Hormones
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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