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Products Details
Product Description
– CBP/EP300-IN-2 is an inhibitor of CBP/EP300 with IC50 values of 1.07 nM and 5.96 nM for CBP/HTRF and Myc, respectively. CBP/EP300-IN-2, example 25, is extracted from patent WO2017205538A1[1].
Web ID
– HY-128761
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C27H29F2N7O2
References
– [1]Patrick Cyr, et al. Pyrazolopyridine derivatives for the treatment of cancer
CAS Number
– 2158265-96-2
Molecular Weight
– 521.56
SMILES
– O=C(N1CCC(N(C2CCOCC2)N=C3C4=CN=CC5=C4C=C(C(F)F)C(C6=CN(C)N=C6)=C5)=C3C1)NC
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
