Download Files:
Products Details
Product Description
– BET-IN-1 is a potent BET inhibitor that has excellent brain penetration and reasonable metabolic stability.
Web ID
– HY-115727
Shipping
– Room temperature
Molecular Formula
– C23H24ClFN4O3S
References
– [1]Bai P, et al. Design, Synthesis, and Evaluation of Thienodiazepine Derivatives as Positron Emission Tomography Imaging Probes for Bromodomain and Extra-Terminal Domain Family Proteins. J Med Chem. 2021 Oct 14;64(19):14745-14756.
CAS Number
– 2727161-43-3
Molecular Weight
– 490.98
SMILES
– ClC1=CC=C(C2=N[C@H](C3=NN=C(N3C4=C2C(C)=C(S4)C)C)CC(OCCOCCF)=O)C=C1
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
