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Product Description
– 4-Methylhistamine (hydrochloride) is a potent, high affinity H4 receptor agonist Ki of 7 nM. 4-Methylhistamine (hydrochloride) displays more than 100-fold selectivity over other human histamine receptor subtypes[1].
Web ID
– HY-W580721A
Shipping
– Room temperature
Molecular Formula
– C6H12ClN3
References
– [1]Lim HD, et.al. Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist. J Pharmacol Exp Ther. 2005 Sep;314(3):1310-21.
CAS Number
– 84103-51-5
Molecular Weight
– 161.63
SMILES
– NCCC1=C(C)N=CN1.[H]Cl
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– 10 mM in DMSO
Target
– Histamine Receptor
Pathway
– GPCR/G Protein, Immunology/Inflammation, Neuronal Signaling
Product type
– Reference compound
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