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Grapiprant
Price range: 48 CAD through 899 CAD
Products Details
Product Description
– Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).
Web ID
– TQ0292
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C26H29N5O3S
References
– Vito VD, et al. Detection and quantification of the selective EP4 receptor antagonist CJ-023423 (grapiprant) in canine plasma by HPLC with spectrofluorimetric detection. J Pharm Biomed Anal. 2016 Jan 25;118:251-8.
CAS Number
– 415903-37-6
Molecular Weight
– C26H29N5O3S
Compound Purity
– 0.9949
SMILES
– CCc1nc2c(C)nc(C)cc2n1-c1ccc(CCNC(=O)NS(=O)(=O)c2ccc(C)cc2)cc1
Pathway
– GPCR/G Protein|||Immunology/Inflammation
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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