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C 21
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Products Details
Product Description
– Selective protein arginine methyltransferase 1 (PRMT1) inhibitor (IC50 = 1.8 μM). Exhibits five-fold selectivity for PRMT1 over PRMT6 and >250-fold selectivity over PRMT3 and CARM1.
Web ID
– TP2041
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C90H161ClN36O24
References
– Obianyo et al (2010) A chloroacetamidine-based inactivator of protein arginine methyltransferase 1: design, synthesis, and in vitro and in vivo evaluation. Chembiochem 11 1219 PMID:
CAS Number
– 1229236-78-5
Molecular Weight
– C90H161ClN36O24
SMILES
– [C@H](CC1=CN=CN1)(C(N[C@H](C(N[C@H](C(N[C@@H]([C@H](C)C)C(O)=O)=O)CCCCN)=O)CCCNC(=N)N)=O)NC([C@@H](NC([C@@H](NC([C@@H](NC(CNC(CNC([C@@H](NC(CNC([C@@H](NC(CNC([C@@H](NC(CNC(CNC([C@@H](NC(CNC([C@@H](NC(CNC([C@@H](NC(C)=O)CO)=O)=O)CCCNC(CCl)=N)=O)=O)CCCCN)=O)=O)=O)CCCCN)=O)=O)CC(C)C)=O)=O)CCCCN)=O)=O)=O)C)=O)CCCCN)=O)CCCNC(=N)N)=O
Product type
– Peptide
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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