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CBP/p300-IN-5
$878
Only 1000 item(s) left in stock.
Products Details
Product Description
– P300/CBP-IN-5 is a potent p300/CBP histone acetyltransferase inhibitor extracted from patent WO2016044770A1, Example 715, has an IC50 of 18.8 nM[1].
Web ID
– HY-100132
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C29H27F5N6O4
References
– [1]Michael Michaelides, et al. Spirocyclic hat inhibitors and methods for their use. WO2016044770A1.
CAS Number
– 1889284-33-6
Molecular Weight
– 618.55
SMILES
– O=C(CN(C1=O)C(N[C@@]21C[C@H](C3=C2C=CC(C4=CN(N=C4)CC(NC)=O)=C3)F)=O)N([C@H](C(F)(F)F)C)CC5=CC=C(C=C5)F
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Acetyltransferase
Isoform
– CBP/p300
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
