GSK-215083

SKU T27455-25 mg Category Small Compound Brand: TargetMol

Price range: 2,432 CAD through 4,000 CAD

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Product Description

– GSK-215083 is a PET radioligand for the 5-HT6 receptor. GSK 215083 is a quinoline based compounds and acts by antagonising the 5-HT6 receptor. GSK-215083 binds to receptors 5-hydroxytrypamine-6 (5HT6) in the striatum and 5-hydroxytryptamine-2A (5HT2A) in the frontal cortex.

Web ID

– T27455

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C20H20FN3O2S

References

– Parker CA, Rabiner EA, Gunn RN, Searle G, Martarello L, Comley RA, Davy M, Wilson AA, Houle S, Mizrahi R, Laruelle M, Cunningham VJ. Human Kinetic Modeling of the 5HT6 PET Radioligand 11C-GSK215083 and Its Utility for Determining Occupancy at Both 5HT6 and 5HT2A Receptors by SB742457 as a Potential Therapeutic Mechanism of Action in Alzheimer Disease. J Nucl Med. 2015 Dec;56(12):1901-9. doi: 10.2967/jnumed.115.162743. Epub 2015 Sep 17. PubMed PMID: 26383152.

CAS Number

– 607742-80-3

Molecular Weight

– C20H20FN3O2S

SMILES

– S(=O)(=O)(C1=CC2=C(C(=CC=C2)N3CCN(C)CC3)N=C1)C4=CC(F)=CC=C4

Pathway

– Others

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

GSK-215083

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