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TRPM8 antagonist 3
$280 – $1,950
Products Details
Product Description
– TRPM8 antagonist 3 is a novel TRPM8 blocker with an IC50 value of 11 nM.
Web ID
– HY-145124
Storage Temperature
– -20°C, 3 years (Powder)
Shipping
– Blue Ice
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C13H12N2O4S
References
– [1]Bianchini G, et al. Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions: A Journey through pKa and LogD Modulation. J Med Chem. 2021 Nov 25;64(22):16820-16837.
CAS Number
– 2102179-29-1
Molecular Weight
– 292.31
Compound Purity
– 99.62
SMILES
– O=C(N1OCCC1)C2=C(O)N=C(C3=C(O)C=CC=C3)S2
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– DMSO : 25 mg/mL (ultrasonic)
Target
– TRP Channel
Pathway
– Membrane Transporter/Ion Channel;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
