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Treprostinil palmitil
SKU
HY-109163-1 mg
Category Reference compound
Tags Endocrinology; Inflammation/Immunology, GPCR/G Protein, Prostaglandin Receptor
$100 – $2,560
Products Details
Product Description
– Treprostinil palmitil (TP) is the proagent of DP1 and EP2 agonist, Treprostinil (UT-15), whose EC50 values were 0.6 and 6.2 nM, respectively. Treprostinil palmitil is a pure proagent and possesses no inherent binding to G-protein coupled receptors including prostanoid receptors[1][2].
Web ID
– HY-109163
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture and light)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C39H66O5
References
– [1]Chapman RW, Corboz MR, Malinin VS, Plaunt AJ, Konicek DM, Li Z, Perkins WR. An overview of the biology of a long-acting inhaled treprostinil prodrug. Pulm Pharmacol Ther. 2020 Dec;65:102002.
CAS Number
– 1706528-83-7
Molecular Weight
– 614.94
Compound Purity
– 99.56
SMILES
– CCCCC[C@H](O)CC[C@@H]1[C@]2([H])[C@@](C[C@H]1O)([H])CC3=C(OCC(OCCCCCCCCCCCCCCCC)=O)C=CC=C3C2
Clinical Information
– Phase 3
Research Area
– Endocrinology; Inflammation/Immunology
Solubility
– DMSO : 200 mg/mL (ultrasonic)
Target
– Prostaglandin Receptor
Isoform
– DP
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.