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Products Details
Product Description
– Tigolaner-d4 is deuterium labeled Tigolaner. Tigolaner is a GABA antagonist that regulates chloride channel. Tigolaner is an antiparasitic agent[1].
Web ID
– HY-109077S
Shipping
– Room temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C21H9D4ClF8N6O
References
– [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.|[2]The use ofstems in the selectionofInternationa Nonproprietary Names(INN)forpharmaceutical substances 2018 (Stem Book2018).
Molecular Weight
– 556.83
SMILES
– O=C(NC1(C#N)C([2H])([2H])C1([2H])[2H])C2=CC(C3=CN(C4=C(C(F)(F)F)C(C(F)(F)C(F)(F)F)=NN4C)N=C3)=CC=C2Cl
Clinical Information
– No Development Reported
Research Area
– Infection; Neurological Disease
Solubility
– 10 mM in DMSO
Target
– GABA Receptor;Isotope-Labeled Compounds;Parasite
Pathway
– Anti-infection;Membrane Transporter/Ion Channel;Neuronal Signaling;Others
Product type
– Isotope-Labeled Compounds
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
