Products Details

Product Description

– Terlakiren (CP-80,794) is an orally active inhibitor of renin. Terlakiren inhibits the efficacy of human renin with an IC50 value of 0.7 nM. Terlakiren has potential applications in hypertension[1].

Web ID

– HY-105205

Shipping

– Room temperature

Molecular Formula

– C31H48N4O7S

References

– [1]Fouda H, et al. Quantitative analysis by high-performance liquid chromatography atmospheric pressure chemical ionization mass spectrometry: The determination of the renin inhibitor CP-80,794 in human serum. J Am Soc Mass Spectrom. 1991 Apr;2(2):164-7.

CAS Number

– 119625-78-4

Molecular Weight

– 620.80

SMILES

– CC(C)OC([C@H](O)[C@@](CC1CCCCC1)([H])NC([C@H](CSC)NC([C@@H](NC(N2CCOCC2)=O)CC3=CC=CC=C3)=O)=O)=O

Clinical Information

– No Development Reported

Research Area

– Cardiovascular Disease

Solubility

– 10 mM in DMSO

Target

– Renin

Pathway

– Metabolic Enzyme/Protease

Product type

– Reference compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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