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Products Details
Product Description
– sst2 Receptor agonist-1 is a potent somatostatin receptor subtype 2 (sst2) agonist with a Ki value of 0.025 nM and a cAMP IC50 value of 4.8 nM. sst2 Receptor agonist-1 can inhibit rat growth hormone (GH) secretion and ocular neovascular lesion formation. Antiangiogenic effect[1].
Web ID
– HY-110161
Shipping
– Room temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C26H25ClN2O2
References
– [1]Wolkenberg SE, et al. Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2. J Med Chem. 2011 Apr 14;54(7):2351-8.
CAS Number
– 1021912-42-4
Molecular Weight
– 432.94
SMILES
– ClC1=CC2=NC=C(C(OCCCN)=C2C=C1C3=CC=CC(O)=C3)C4=CC(C)=CC(C)=C4
Clinical Information
– No Development Reported
Research Area
– Endocrinology; Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– Somatostatin Receptor
Isoform
– SSTR2
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
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