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Products Details
Product Description
– sPLA2-X Inhibitor 31 is a selective secreted phospholipase A2 type X (sPLA2-X) inhibitor with IC50s of 26 nM, 310 nM, and 2230 nM for sPLA2-X, sPLA2-IIa, and sPLA2-V, respectively[1].
Web ID
– HY-112605
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C19H15F3N2O4
References
– [1]Knerr L, et al. Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A2 Type X(sPLA2-X) Inhibitors. ACS Med Chem Lett. 2018 Jun 23;9(7):594-599.
CAS Number
– 2241025-50-1
Molecular Weight
– 392.33
SMILES
– FC(F)(F)OC1=CC=C(C=C(C(N)=O)N2C3=CC(CCC(O)=O)=CC=C3)C2=C1
Clinical Information
– No Development Reported
Research Area
– Cardiovascular Disease
Solubility
– 10 mM in DMSO
Target
– Phospholipase
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
