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SORT-PGRN interaction inhibitor 1
SKU
HY-115213-100 mg
Category Reference compound
Tags GPCR/G Protein;Neuronal Signaling, Neurological Disease, Neurotensin Receptor
$50 – $90
Products Details
Product Description
– SORT-PGRN interaction inhibitor 1 is a potent inhibitor of the sortilin-progranulin interaction with an IC50 of 2 μM[1].
Web ID
– HY-115213
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C15H18N2O2
References
– [1]Shawn J Stachel, et al. Identification of potent inhibitors of the sortilin-progranulin interaction. Bioorg Med Chem Lett. 2020 Sep 1;30(17):127403.
CAS Number
– 100957-85-5
Molecular Weight
– 258.32
Compound Purity
– 98.94
SMILES
– O=C(C1=CC(C(C)(C)C)=NN1CC2=CC=CC=C2)O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– Neurotensin Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.