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SNT-207707
$300 – $4,100
Products Details
Product Description
– SNT-207707 is a selective, potent and orally active melanocortin MC-4 receptor antagonist with an IC50 of 8 nM (binding) and 5 nM (function) on the MC-4 receptor.
Web ID
– HY-11029
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C32H44ClN5O
References
– [1]Weyermann P, et al. Orally available selective melanocortin-4 receptor antagonists stimulate food intake and reduce cancer-induced cachexia in mice. PLoS One. 2009;4(3):e4774.
CAS Number
– 1064662-40-3
Molecular Weight
– 550.18
Compound Purity
– 99.51
SMILES
– O=C(C1=CN2C(C=C1)=NC(C3=CC=C(C#N)C=C3)=C2CCCN4CCCC4)N(CCC(C)C)CCC(C)C.Cl
Clinical Information
– No Development Reported
Research Area
– Cancer; Metabolic Disease; Endocrinology
Solubility
– DMSO : ≥ 250 mg/mL
Target
– Melanocortin Receptor
Isoform
– MC4R
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
