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Sheng Gelieting
SKU
HY-148190-Get quote
Category Reference compound
Tags Dipeptidyl Peptidase, Endocrinology, Metabolic Enzyme/Protease
Products Details
Product Description
– Sheng Gelieting (CGT-8012) is a dipeptidy peptidase-IV enzyme (DP-IV) inhibitor. Sheng Gelieting has great DP-IV inhibition activity with an IC50 value of 87 nM. Sheng Gelieting can be used for curing or preventing diseases relevant to the dipeptidy peptidase-IV enzyme, such as the diabetes, particularly the II-type diabete[1].
Web ID
– HY-148190
Shipping
– Room temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C17H16F6N4O
References
– [1]Qiang Yu, et al. Beta-amino tetrahydropyrazine, tetrahydropyrimidine and tetrahydropyridine used as dipeptidy peptidase inhibitors for curing or preventing diabetes. Patent. CN101899047A.
CAS Number
– 1152810-23-5
Molecular Weight
– 406.33
SMILES
– FC(F)(C1=NC=C2N1CCN(C(C[C@H](N)CC3=C(C=C(C(F)=C3)F)F)=O)C2)F
Clinical Information
– No Development Reported
Research Area
– Endocrinology
Solubility
– 10 mM in DMSO
Target
– Dipeptidyl Peptidase
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
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