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Setastine
SKU
HY-119832-Get quote
Category Reference compound
Tags GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling, Histamine Receptor, Inflammation/Immunology
Products Details
Product Description
– Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<.
Web ID
– HY-119832
Shipping
– Room temperature
Molecular Formula
– C22H28ClNO
References
– [1]Németh, A., & Huszti, Z. (1988). The effect of a new antihistamine drug, Loderix® (EGIS-2062), on stimulus-evoked histamine release from rat peritoneal mast cells. Agents and Actions, 23(3-4), 194–197.
CAS Number
– 64294-95-7
Molecular Weight
– 357.92
SMILES
– CC(C1=CC=C(C=C1)Cl)(OCCN2CCCCCC2)C3=CC=CC=C3
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Histamine Receptor
Pathway
– GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.